RESULT OF DRUG
Total records: 1 Records
 
Record No:1
| ACCESS NO | 4148 |
| DRUG_NAME | Molidustat |
| DRUG_BANK_ID | DB15642 |
| PUBCHEM_ID | 59603622 (CID) |
| STATUS | Research |
| IC50_EC50 | 450.0 nM (IC50 value) |
| ASSAY_ORGANISM | Human |
| ASSAY_DESCRIPTION | Inhibition of recombinant human HIF-PHD3 expressed in baculovirus-infected Sf9 cells using biotin labelled DLDLEMLAPYIPMDDDFQL as substrate preincubated for 60 mins followed by substrate addition measured after 60 mins by TR-FRET assay |
| TARGET_ORGANISM | Human |
| OFF_TARGET | - |
| PMID | 29712435 |