RESULT OF DRUG
Total records: 1 Records
 
Record No:1
| ACCESS NO | 4203 |
| DRUG_NAME | Galunisertib |
| DRUG_BANK_ID | DB11911 |
| PUBCHEM_ID | 10090485 (CID) |
| STATUS | Investigational (Phase II) |
| IC50_EC50 | 51.0 nM (IC50 value) |
| ASSAY_ORGANISM | Human |
| ASSAY_DESCRIPTION | Inhibition of human ALK5 expressed in Sf9 insect cells using casein as substrate in presence of [gamma-33P]ATP |
| TARGET_ORGANISM | Human |
| OFF_TARGET | - |
| PMID | 28135685 |